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4

抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T0442 Bucetin

3-Hydroxy-p-butyrophenetidide,布西丁,羟丁酰胺苯醚

Others Others
Bucetin (3-Hydroxy-p-butyrophenetidide) 是解热化合物,可用于研究疼痛的缓解。
T1386 Phenazopyridine hydrochloride

Urodine,Pyridium,Phenazopyridine HCl,盐酸非那吡啶

Sodium Channel Membrane transporter/Ion channel
Phenazopyridine hydrochloride (Pyridium) 是一种具有局部止痛作用的化学物质,常被用于缓解手术、损伤尿道及尿路感染引起的疼痛、刺激、不适和尿急。
T15300 Fluorofenidone

AKF-PD

Others Others
Fluorofenidone (AKF-PD) 是 AMR69 的类似物,抗纤维化活性与 AMR69相同,但 Fluorofenidone 的毒性更低,半衰期长。它部分通过 PI3K/Akt 信号通路抑制 NADPH 氧化酶和细胞外基质 (ECM) 的沉积,能够减少肾间质纤维化的发生。
T35893 rac-1,2-bis-Palmitoyl-3-chloropropanediol

rac-1,2-bis-Palmitoyl-3-chloropropanediol is a 3-monochloropropane-1,2-diol (3-MCPD) ester.1It has been found as a contaminant in edible olive oils, with the lowest and highest concentrations in extra virgin and olive pomace oils, respectively.rac-1,2-bis-Palmitoyl-3-chloropropanediol has also been found in cottonseed and palm oils, as well as in shortening.2It induces renal tubular necrosis and a decrease in spermatids, but no gross pathological changes, in mice.3 1.Hung, W.-C., Peng, G.-J., Ts...

化合物

Bucetin
Cat.No: T0442
Synonym: 3-Hydroxy-p-butyrophenetidide,布西丁,羟丁酰胺苯醚
Target: Others
Phenazopyridine hydrochloride
Cat.No: T1386
Synonym: Urodine,Pyridium,Phenazopyridine HCl,盐酸非那吡啶
Target: Sodium Channel
Fluorofenidone
Cat.No: T15300
Synonym: AKF-PD
Target: Others
rac-1,2-bis-Palmitoyl-3-chloropropanediol
Cat.No: T35893
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5669 Citric acid monohydrate

Others Others
Citric acid monohydrate 是一种存在于柑橘类水果中的三羧酸。柠檬酸因其抗氧化特性而被用作药物制剂中的赋形剂。它保持活性成分的稳定性并用作防腐剂。
T5S0636 Citric acid

柠檬酸,Citro,Citretten

Apoptosis; Others; Endogenous Metabolite; Antibacterial; Antibiotic Apoptosis; Metabolism; Microbiology/Virology; Others
Citric acid (Citro) 是柑橘类水果中发现的弱有机三羧酸。柠檬酸是食品添加剂和天然防腐剂。
T81629 OAT1/3-IN-2

OAT1/3-IN-2(化合物8)是一种针对OAT1和OAT3的双重抑制剂。该化合物能够以10 μM的浓度逆转Cys-Hg对HEK-OAT1细胞的毒害作用,并可能对肾脏具有保护效应。OAT1/3-IN-2适用于研究汞导致的肾脏损伤。
T81630 OAT1/3-IN-1

OAT1/3-IN-1(化合物7)是针对OAT1和OAT3的双重抑制剂。该化合物能逆转Cys-Hg(10 μM)对HEK-OAT1细胞引起的毒害,表明其对肾脏有潜在的保护效应。OAT1/3-IN-1适合用于探究汞引起的肾脏损伤机制研究。

天然产物

Citric acid monohydrate
Cat.No: T5669
Synonym:
Target: Others
Citric acid
Cat.No: T5S0636
Synonym: 柠檬酸,Citro,Citretten
Target: Apoptosis, Others, Endogenous Metabolite, Antibacterial, Antibiotic
OAT1/3-IN-2
Cat.No: T81629
Synonym:
Target:
OAT1/3-IN-1
Cat.No: T81630
Synonym:
Target:
TargetMol Loading
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